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Synthesis and Biological Evaluation of New Quinoxaline Derivatives of ICF01012 as Melanoma-Targeting Probes
Emmanuel Moreau
,
Radhia El Aissi
,
Jianrong Liu
,
Sophie Besse
,
Damien Canitrot
et al.
Journal articles
hal-01677548v1
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Design, Synthesis, Biological Evaluation, and Structure–Activity Relationships of Substituted Phenyl 4-(2-Oxoimidazolidin-1-yl)benzenesulfonates as New Tubulin Inhibitors Mimicking Combretastatin A-4
Emmanuel Moreau
,
Sébastien Fortin
,
Lianhu Wei
,
Jacques Lacroix
,
Marie-France Côté
et al.
Journal articles
hal-01677554v1
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A Photochemical Approach to Pyridopyrroloquinoline Derivatives as New Potential Anticancer Agents
Pierre-Jean Aragon
,
Ange-Désiré Yapi
,
Frédéric Pinguet
,
Jean-Michel Chezal
,
Jean-Claude Teulade
et al.
Journal articles
hal-02384520v1
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N-Phenyl-N′-(2-chloroethyl)ureas (CEU) as potential antineoplastic agents. Part 2: Role of ω-hydroxyl group in the covalent binding to β-tubulin
Emmanuel Moreau
,
Sébastien Fortin
,
Alexandre Patenaude
,
Michel Desjardins
,
Jacques Lacroix
et al.
Journal articles
hal-01677583v1
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A comparative molecular field and comparative molecular similarity indices analyses (CoMFA and CoMSIA) of N-phenyl-N′-(2-chloroethyl)ureas targeting the colchicine-binding site as anticancer agents
Emmanuel Moreau
,
Sébastien Fortin
,
Philippe Labrie
,
Lianhu Wei
,
Lakshmi P Kotra
et al.
Journal articles
hal-01677579v1
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Mechanism of action of N-phenyl-N′-(2-chloroethyl)ureas in the colchicine-binding site at the interface between α- and β-tubulin
Emmanuel Moreau
,
Sébastien Fortin
,
Lianhu Wei
,
Philippe Labrie
,
Éric Petitclerc
et al.
Journal articles
hal-01677570v1
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A Novel HPLC Method for Direct Detection of Nitric Oxide Scavengers from Complex Plant Matrices and Its Application to Aloysia triphylla Leaves
Didier Fraisse
,
Alexandra Degerine-Roussel
,
Alexis Bred
,
Samba Ndoye
,
Magali Vivier
et al.
Journal articles
hal-01873226v1
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Inhibition profiles of mono- and polyvalent FimH antagonists against 10 different Escherichia coli strains
T. Chalopin
,
Y. Brissonnet
,
Adeline Sivignon
,
D. Deniaud
,
L. Cremet
et al.
Journal articles
hal-01931394v1
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Elaboration et caractérisation d’un hybride organominéral à base de polycaprolactone et de bioverre sous forme de mousse macroporeuse pour la régénération osseuse
Cédric Bossard
Chimie thérapeutique. Université Clermont Auvergne [2017-2020], 2018. Français. ⟨NNT : 2018CLFAC068⟩
Theses
tel-02128441v1
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Expeditious Synthesis of the Topoisomerase I Inhibitors Isoindolo[2,1-b]isoquinolin-7(5H)-one and the Alkaloid Rosettacin Based on Aryl Radical Cyclization of Enamide Generated by Using N-Acyliminium Chemistry
Ata Martin Lawson
,
Lahssen El Blidi
,
Aurélie Namoune
,
Alexandre Bridoux
,
Vijaykumar Nimbarte
et al.
Journal articles
hal-02332633v1
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Imidazonaphthyridine systems (part 2): Functionalization of the phenyl ring linked to the pyridine pharmacophore and its replacement by a pyridinone ring produces intriguing differences in cytocidal activity
Emmanuel Moreau
,
Nicolas Masurier
,
Eric Debiton
,
Alicia Jacquemet
,
Antoine Bussière
et al.
Journal articles
hal-01677549v1
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Heteropolysaccharides from S. cerevisiae show anti-adhesive properties against E. coli associated with Crohn’s disease
Adeline Sivignon
,
Shin-Yi Yu
,
Nathalie Ballet
,
Pascal Vandekerckove
,
Nicolas Barnich
et al.
Journal articles
hal-03373401v1
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Linker structure-activity relationships in fluorodeoxyglucose chlorambucil conjugates for tumor-targeted chemotherapy
Valérie Weber
,
Mostafa El Hilali
,
Bastien Reux
,
Eric Debiton
,
Fernand Leal
et al.
Journal articles
hal-01677115v1
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Characterization of the Covalent Binding of N-Phenyl-N'-(2-chloroethyl)ureas to -Tubulin: Importance of Glu198 in Microtubule Stability
Emmanuel Moreau
,
S. Fortin
,
B. Bouchon
,
C. Chambon
,
J. Lacroix
et al.
Journal articles
hal-01677562v1
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N-Substituted 4-aminobenzamides (procainamide analogs): an assessment of multiple cellular effects vis-a-vis ion trapping
Emmanuel Moreau
,
G. Morissette
Journal articles
hal-01677587v1
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Optimized N-phenyl-N′-(2-chloroethyl)ureas as potential antineoplastic agents: Synthesis and growth inhibition activity
Emmanuel Moreau
,
Sébastien Fortin
,
Michel Desjardins
,
Jean L C Rousseau
,
Eric Petitclerc
et al.
Journal articles
hal-01677590v1
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Heterocyclization of Functionalized Vinylic Derivatives of Imidazo[1,2- a ]pyridines
Emmanuel Moreau
,
Jean Chezal
,
Gregory Delmas
,
Alain Gueiffier
,
Yves Blache
et al.
Journal articles
istex
hal-01677665v1
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Black mamba venom peptides target acid-sensing ion channels to abolish pain
Sylvie Diochot
,
Anne Baron
,
Miguel Salinas
,
Dominique Douguet
,
Sabine Scarzello
et al.
Journal articles
istex
hal-02115775v1
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Current Opinion on Chitosan and its Derivatives: Biological Impact in Antimicrobial Applications From Nature to Chitosan and It Derivatives: How it is Working?
Cédric Delattre
Journal articles
hal-01657856v1
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Effect of proteases against biofilms of Staphylococcus aureus and Staphylococcus epidermidis
Pierre-Henri Elchinger
,
C. Delattre
,
S. Faure
,
O. Roy
,
S. Badel
et al.
Journal articles
hal-01081362v1
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Synthesis of Polyfused Heterocycle Derivatives Containing the Dipyridoimidazole Core by Friedländer’s Reaction: Access to Analogs of Ellipticine
Emmanuel Moreau
,
Jean-Claude Teulade
,
Nicolas Desbois
,
Jean-Michel J.-M. Chezal
,
Florence Fauvelle
et al.
Journal articles
hal-01677674v1
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Chemo-enzymatic synthesis of a series of 2,4-syn-functionalized (S)-glutamate analogues: new insight into the structure-activity relation of ionotropic glutamate receptor subtypes 5, 6, and 7.
Emmanuelle Sagot
,
Darryl S. Pickering
,
Xiasui Pu
,
Michelle Umberti
,
Tine B. Stensbol
et al.
Journal of Medicinal Chemistry, 2008, 51, pp.4093-4103
Journal articles
hal-00323861v1
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Pharmacological characterization of (4R)-alkyl glutamate analogues at the ionotropic glutamate receptors - Focus on subtypes iGluR5-7
Lennart Bunch
,
Thierry Gefflaut
,
Sébastien Alaux
,
Emmanuelle Sagot
,
Brigitte Nielsen
et al.
European Journal of Pharmacology, 2009, 609, pp.1-4
Journal articles
hal-00376953v1
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Synthesis, in vitro antiproliferative activities, and Chk1 inhibitory properties of pyrrolo[3,4-a]carbazole-1,3-diones, pyrrolo[3,4-c]carbazole-1,3-diones, and 2-aminopyridazino[3,4-a]pyrrolo[3,4-c]carbazole-1,3,4,7-tetraone
Elisabeth Conchon
,
Fabrice Anizon
,
Bettina Aboab
,
Roy Golsteyn
,
Stéphane Leonce
et al.
European Journal of Medicinal Chemistry, 2008, 43, pp.282-292
Journal articles
hal-00255899v1
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Metabolic and Anti-Inflammatory Protective Properties of Human Enriched Serum Following Artichoke Leaf Extract Absorption: Results from an Innovative Ex Vivo Clinical Trial
Fabien Wauquier
,
Line Boutin-Wittrant
,
Aurélien Viret
,
Laure Guilhaudis
,
Hassan Oulyadi
et al.
Journal articles
hal-03326084v1
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Gliotransmission and Brain Glucose Sensing: Critical Role of Endozepines
Damien Lanfray
,
Sébastien Arthaud
,
Johanne Ouellet
,
Vincent Compère
,
Jean-Luc Do Rego
et al.
Journal articles
hal-01962799v1
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Involvement of the Acyl-CoA binding domain containing 7 in the control of food intake and energy expenditure in mice
Damien Lanfray
,
Alexandre Caron
,
Marie-Claude Roy
,
Mathieu Laplante
,
Fabrice Morin
et al.
Journal articles
hal-01962802v1
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Massive Cell Vacuolization Induced by Organic Amines Such as Procainamide
Emmanuel Moreau
,
G. Morissette
Journal articles
hal-01677592v1
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Benefits of the ipowder® extraction process applied to Melissa officinalis L.: improvement of antioxidant activity and in vitro gastro-intestinal release profile of rosmarinic acid
Valérie Bardot
,
Anaïs Escalon
,
Isabelle Ripoche
,
Sylvain Denis
,
Monique Alric
et al.
Journal articles
hal-02441644v1
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Novel imidazo[1,2-a]naphthyridinic systems (part 1): Synthesis, antiproliferative and DNA-intercalating activities
Emmanuel Moreau
,
Mounir Andaloussi
,
Nicolas Masurier
,
Jacques Lacroix
,
René C Gaudreault
et al.
Journal articles
istex
hal-01677576v1
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