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Synthesis and Biological Evaluation of New Quinoxaline Derivatives of ICF01012 as Melanoma-Targeting Probes
Emmanuel Moreau
,
Radhia El Aissi
,
Jianrong Liu
,
Sophie Besse
,
Damien Canitrot
et al.
Journal articles
hal-01677548v1
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Design, Synthesis, Biological Evaluation, and Structure–Activity Relationships of Substituted Phenyl 4-(2-Oxoimidazolidin-1-yl)benzenesulfonates as New Tubulin Inhibitors Mimicking Combretastatin A-4
Emmanuel Moreau
,
Sébastien Fortin
,
Lianhu Wei
,
Jacques Lacroix
,
Marie-France Côté
et al.
Journal articles
hal-01677554v1
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(2 R ,3 S )-2-Ammonio-3-hydroxy-3-(4-nitrophenyl)propanoic acid chloride monohydrate
Vincent Gaumet
,
Valérie Weber
,
Valery Zaitsev
,
Michel Madesclaire
Journal articles
hal-02885166v1
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Development of a freeze-dried kit formulation for the preparation of 99m Tc-NTP 15-5, a radiotracer for scintigraphic imaging of proteoglycans
Aurélien Vidal
,
Vincent Gaumet
,
Marie-Josephe Galmier
,
Sophie Besse
,
Fernand Leal
et al.
Journal articles
hal-01961372v1
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A comparative molecular field and comparative molecular similarity indices analyses (CoMFA and CoMSIA) of N-phenyl-N′-(2-chloroethyl)ureas targeting the colchicine-binding site as anticancer agents
Emmanuel Moreau
,
Sébastien Fortin
,
Philippe Labrie
,
Lianhu Wei
,
Lakshmi P Kotra
et al.
Journal articles
hal-01677579v1
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Mechanism of action of N-phenyl-N′-(2-chloroethyl)ureas in the colchicine-binding site at the interface between α- and β-tubulin
Emmanuel Moreau
,
Sébastien Fortin
,
Lianhu Wei
,
Philippe Labrie
,
Éric Petitclerc
et al.
Journal articles
hal-01677570v1
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N-Phenyl-N′-(2-chloroethyl)ureas (CEU) as potential antineoplastic agents. Part 2: Role of ω-hydroxyl group in the covalent binding to β-tubulin
Emmanuel Moreau
,
Sébastien Fortin
,
Alexandre Patenaude
,
Michel Desjardins
,
Jacques Lacroix
et al.
Journal articles
hal-01677583v1
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[(2 R ,3 R )-3-(4-Nitrophenyl)aziridin-2-yl]methanol monohydrate
Vincent Gaumet
,
C. Denis
,
F. Leal
,
M. Madesclaire
,
V.P. Zaitsev
et al.
Journal articles
hal-02885206v1
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Imidazonaphthyridine systems (part 2): Functionalization of the phenyl ring linked to the pyridine pharmacophore and its replacement by a pyridinone ring produces intriguing differences in cytocidal activity
Emmanuel Moreau
,
Nicolas Masurier
,
Eric Debiton
,
Alicia Jacquemet
,
Antoine Bussière
et al.
Journal articles
hal-01677549v1
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Macrocyclic complexes, their process of preparation and use as PET imaging agents
Vincent Gaumet
,
Claire Denis
,
Aurélien Vidal
,
Philippe Auzeloux
,
Jean-Claude Madelmont
et al.
France, Patent n° : WO2016016272 (A1). 2016
Patents
hal-02885526v1
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Massive Cell Vacuolization Induced by Organic Amines Such as Procainamide
Emmanuel Moreau
,
G. Morissette
Journal articles
hal-01677592v1
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Novel imidazo[1,2-a]naphthyridinic systems (part 1): Synthesis, antiproliferative and DNA-intercalating activities
Emmanuel Moreau
,
Mounir Andaloussi
,
Nicolas Masurier
,
Jacques Lacroix
,
René C Gaudreault
et al.
Journal articles
istex
hal-01677576v1
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Enhancement of cationic conductivity in some heptafluorozirconates due to a paddle-wheel mechanism
Vincent Gaumet
,
C. Latouche
,
D Avignant
,
J. Dupuis
Journal articles
istex
hal-02883790v1
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2,2′-Bipyrimidine as a Building Block for the Design of Emissive Conjugated Polymers for Hybrid LED Lighting
Qiqiao Lin
,
Xiaoguang Huang
,
Sasikumar Ramachandran
,
Xinyang Wang
,
Rachod Boonsin
et al.
Journal articles
hal-03086161v1
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Stereoselective synthesis of (E)-N,N-diethyl-3-(imidazo[1,2-a]pyrid-2-yl)-2-(phenylsulfonyl)propenamide
S. Céard
,
D. Roche
,
Vincent Gaumet
,
D. Gardette
,
J. Metin
et al.
Journal articles
istex
hal-02885118v1
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Synthesis of carbamoylpyridine and imidazo[1,5-a]pyridin-1,3-diones via ortho-acetalhydantoin intermediates
Jean Chezal
,
Emmanuel Moreau
,
Nicolas Desbois
,
Yves Blache
,
Olivier Chavignon
et al.
Journal articles
istex
hal-01677650v1
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Synthesis and antiviral activity of an imidazo[1,2-a]pyrrolo[2,3-c]pyridine series against the bovine viral diarrhea virus
Emmanuel Moreau
,
Jean-Michel J.-M. Chezal
,
Jan Paeshuyse
,
Vincent Gaumet
,
Damien Canitrot
et al.
Journal articles
istex
hal-01677567v1
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New Opportunities with the Duff Reaction
Emmanuel Moreau
,
Nicolas Masurier
,
Claire Lartigue
,
Vincent Gaumet
,
Jean-Michel J.-M. Chezal
et al.
Journal articles
istex
hal-01677572v1
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Synthesis and in vitro evaluation of new fluorinated quinoline derivatives with high affinity for PDE5: Towards the development of new PET neuroimaging probes
Jianrong Liu
,
Aurelie Maisonial-Besset
,
Barbara Wenzel
,
Damien Canitrot
,
Ariane Baufond
et al.
Journal articles
hal-01671041v1
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Melanoma-targeted delivery system (part 1): Design, synthesis and evaluation of releasable disulfide drug by glutathione
Emmanuel Moreau
,
Radhia El Aissi
,
Jean-Michel J.-M. Chezal
,
Sébastien Tarrit
,
Olivier Chavignon
et al.
Journal articles
hal-01677547v1
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Efficient synthesis of novel dipyridoimidazoles and pyrido[1′,2′;1,2]imidazo[4,5-d]pyridazine derivatives
Emmanuel Moreau
,
Jean Chezal
,
Olivier Chavignon
,
Claire Lartigue
,
Yves Blache
et al.
Journal articles
istex
hal-01677655v1
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Efficient Synthesis of New Polyfunctionalized Thiadiazaacenaphthylenes from Imidazo[1,2-a]pyridines
Emmanuel Moreau
,
Jean-Claude Teulade
,
Jean-Michel J.-M. Chezal
,
Caroline Dechambre
,
Damien Canitrot
et al.
Journal articles
hal-01677680v1
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N-Phenyl-N′-(2-chloroethyl)urea analogues of combretastatin A-4: Is the N-phenyl-N′-(2-chloroethyl)urea pharmacophore mimicking the trimethoxy phenyl moiety?
Emmanuel Moreau
,
Sébastien Fortin
,
Jacques Lacroix
,
Jean-Claude Teulade
,
Alexandre Patenaude
et al.
Journal articles
hal-01677582v1
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Synthesis, antiproliferative activity evaluation and structure–activity relationships of novel aromatic urea and amide analogues of N-phenyl-N′-(2-chloroethyl)ureas
Emmanuel Moreau
,
Sébastien Fortin
,
Jacques Lacroix
,
Marie-France Côté
,
Éric Petitclerc
et al.
Journal articles
hal-01677564v1
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Characterization of the Covalent Binding of N-Phenyl-N'-(2-chloroethyl)ureas to -Tubulin: Importance of Glu198 in Microtubule Stability
Emmanuel Moreau
,
S. Fortin
,
B. Bouchon
,
C. Chambon
,
J. Lacroix
et al.
Journal articles
hal-01677562v1
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Optimized N-phenyl-N′-(2-chloroethyl)ureas as potential antineoplastic agents: Synthesis and growth inhibition activity
Emmanuel Moreau
,
Sébastien Fortin
,
Michel Desjardins
,
Jean L C Rousseau
,
Eric Petitclerc
et al.
Journal articles
hal-01677590v1
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Heterocyclization of Functionalized Vinylic Derivatives of Imidazo[1,2- a ]pyridines
Emmanuel Moreau
,
Jean Chezal
,
Gregory Delmas
,
Alain Gueiffier
,
Yves Blache
et al.
Journal articles
istex
hal-01677665v1
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Synthesis of Polyfused Heterocycle Derivatives Containing the Dipyridoimidazole Core by Friedländer’s Reaction: Access to Analogs of Ellipticine
Emmanuel Moreau
,
Jean-Claude Teulade
,
Nicolas Desbois
,
Jean-Michel J.-M. Chezal
,
Florence Fauvelle
et al.
Journal articles
hal-01677674v1
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N-Heterocyclic Pyridylmethylamines: Synthesis, Complexation, Molecular Structure, and Application to Asymmetric Suzuki–Miyaura and Oxidative Coupling Reactions
Guillaume Grach
,
Grégory Pieters
,
Aurelia Dinut
,
Vincent Terrasson
,
Raouf Medimagh
et al.
Journal articles
hal-02194706v1
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X-ray structural analysis of (1R,2R,4S,5S,8S)-2,8-bis(4-chlorophenyl)-4-(4-nitrophenyl)-1-aza-3,7-dioxabicyclo[3,3,0]octane
M. Madesclaire
,
P. Coudert
,
Vincent Gaumet
,
V. Zaitsev
,
J. Zaitseva
et al.
Journal articles
istex
hal-02885161v1
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